SCHEMBL2861257

SCHEMBL2861257

Cc1ccccc1C(=O)C#CC(=O)NC1CCN(c2nc(C)c(C)s2)C1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.37
BTK Q06187 2/20 0.37
PAK1 Q13153 1/20 0.36
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36
POLB P06746 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
SMPD3 Q9NY59 1/20 0.35
DRD4 P21917 2/20 0.35
ACKR3 P25106 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35
CHRM1 P11229 1/20 0.35
ALOX15 P16050 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2855060 0.86 ALDH1A1 (0.43) SMN1; SMN2BTKPAK1POLBKDM4E
SCHEMBL974372 0.85 SMPD3 (0.36) BTKSMPD3DRD4ACKR3NPC1
SCHEMBL2856121 0.85 PAK1 (0.40) SMN1; SMN2BTKPAK1POLBACKR3
SCHEMBL2863170 0.84 PPARG (0.36) SMN1; SMN2BTKPAK1CCNE1CDK2
SCHEMBL2854730 0.83 CTSB (0.37) SMN1; SMN2BTKPAK1POLBACKR3
SCHEMBL973992 0.83 BTK (0.45) BTKSMPD3DRD4NPC1RAB9A
SCHEMBL2858043 0.83 CCNE1 (0.40) SMN1; SMN2BTKCCNE1CDK2NPC1
SCHEMBL974402 0.80 BTK (0.37) BTKCCNE1CDK2SMPD3DRD4
SCHEMBL974290 0.79 BTK (0.38) SMN1; SMN2BTKSMPD3ACKR3NPC1
SCHEMBL973986 0.79 SMPD3 (0.41) BTKSMPD3DRD4NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968957-B1 SUBSTITUTED THIAZOLES AND THEIR USE FOR PRODUCING DRUGS GRUENENTHAL GMBH (DE) 2010-01-20 EP claimed