SCHEMBL28559152

SCHEMBL28559152

Cn1ccc(-c2cncc(-c3ccc(N4CCCC4=O)cc3)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 2/20 0.43
CDK8 P49336 2/20 0.43
CHEK1 O14757 1/20 0.42
ALDH1A1 P00352 1/20 0.42
NPC1 O15118 1/20 0.42
SYK P43405 3/20 0.41
CYP11B2 P19099 5/20 0.41
CYP11B1 P15538 4/20 0.41
HPGD P15428 1/20 0.41
BMPR1B O00238 1/20 0.40
BMPR1A P36894 1/20 0.40
TGFBR1 P36897 1/20 0.40
ACVRL1 P37023 1/20 0.40
ACVR1 Q04771 1/20 0.40
BRD4 O60885 1/20 0.39
BRDT Q58F21 1/20 0.39
IP6K1 Q92551 1/20 0.39
IP6K3 Q96PC2 1/20 0.39
IP6K2 Q9UHH9 1/20 0.39
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22554035 0.85 BMPR1B (0.53) CCNCCDK8CHEK1ALDH1A1NPC1
SCHEMBL22553833 0.84 SYK (0.42) CCNCCDK8CHEK1ALDH1A1NPC1
SCHEMBL28560413 0.82 SYK (0.45) CCNCCDK8CHEK1ALDH1A1NPC1
SCHEMBL28912924 0.82 CYP11B2 (0.45) CCNCCDK8CHEK1ALDH1A1NPC1
SCHEMBL28563345 0.82 NPC1 (0.40) CCNCCDK8ALDH1A1NPC1SYK
SCHEMBL28558370 0.82 NPC1 (0.40) CCNCCDK8CHEK1ALDH1A1NPC1
SCHEMBL28557029 0.82 ACVRL1 (0.40) CCNCCDK8ALDH1A1NPC1SYK
SCHEMBL22553727 0.82 ALDH1A1 (0.48) CHEK1ALDH1A1NPC1CYP11B2CYP11B1
SCHEMBL30730791 0.82 ALDH1A1 (0.48) CHEK1ALDH1A1NPC1CYP11B2CYP11B1
SCHEMBL28553386 0.80 GAA (0.46) CCNCCDK8ALDH1A1NPC1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN claimed
CN-112088157-A Aryl-bipyridine amine derivatives as phosphoinositide kinase inhibitors 拉文纳制药公司 2020-12-15 CN claimed
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN disclosed
CN-112088157-A Aryl-bipyridine amine derivatives as phosphoinositide kinase inhibitors 拉文纳制药公司 2020-12-15 CN disclosed