SCHEMBL28564433

SCHEMBL28564433

NC(=O)Oc1nc2c(Br)cc(F)c(F)c2s1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK4 O00444 1/20 0.30
CHEK1 O14757 1/20 0.30
AURKA O14965 1/20 0.30
DAPK3 O43293 1/20 0.30
PAK4 O96013 1/20 0.30
CHEK2 O96017 1/20 0.30
LCK P06239 1/20 0.30
CDK1 P06493 1/20 0.30
LYN P07948 1/20 0.30
PIM1 P11309 1/20 0.30
FGFR1 P11362 1/20 0.30
PRKACA P17612 1/20 0.30
FLT1 P17948 1/20 0.30
FGFR3 P22607 1/20 0.30
RPS6KB1 P23443 1/20 0.30
CDK2 P24941 1/20 0.30
MARK3 P27448 1/20 0.30
MAPK1 P28482 1/20 0.30
AKT1 P31749 1/20 0.30
FLT4 P35916 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21839593 0.72 NPC1 (0.39)
SCHEMBL21839495 0.72 ALDH1A1 (0.51) MAPK1
SCHEMBL28575299 0.71 PIM1 (0.33) PIM1
SCHEMBL21901455 0.68 LCK (0.49) LCK
SCHEMBL28564366 0.67 MAPT (0.39) LIMK1DYRK1A
SCHEMBL28902824 0.66 CLK1 (0.31) DYRK1A
SCHEMBL27209845 0.65 PDGFRB (0.31) KDR
SCHEMBL28782049 0.65 NPC1 (0.34) DYRK1A
SCHEMBL25368842 0.64 ALDH1A1 (0.32)
SCHEMBL17796987 0.63 SLC1A3 (0.38) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112805281-B KRAS G12C inhibitors 伊莱利利公司 2022-05-10 CN disclosed
CN-112805281-A KRAS G12C inhibitors 伊莱利利公司 2021-05-14 CN disclosed