SCHEMBL28902824

SCHEMBL28902824

NC(=O)Oc1nc2c(O)c(F)ccc2s1

nearest known ligand 0.31

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 1/20 0.31
DYRK1A Q13627 1/20 0.31
DYRK1B Q9Y463 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B1 P14061 2/20 0.31
HSD17B2 P37059 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28575299 0.77 PIM1 (0.33)
SCHEMBL28902795 0.76 CA2 (0.37)
SCHEMBL30231115 0.76 CA2 (0.37)
SCHEMBL29031079 0.73 PTGS2 (0.32)
SCHEMBL30231203 0.73 SMN1; SMN2 (0.58) SMN1; SMN2
SCHEMBL28902805 0.73 SMN1; SMN2 (0.58) SMN1; SMN2
SCHEMBL28782049 0.72 NPC1 (0.34) DYRK1A
SCHEMBL30622711 0.72 ALDH1A1 (0.53) SMN1; SMN2
SCHEMBL28564366 0.72 MAPT (0.39) DYRK1ASMN1; SMN2
SCHEMBL28400513 0.72 ALDH1A1 (0.53) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116390923-A Heterocyclic derivative and preparation method and application thereof 浙江海正药业股份有限公司 2023-07-04 CN disclosed
CN-115403575-A Heteroaromatic ring derivative and preparation method and application thereof 浙江海正药业股份有限公司 2022-11-29 CN disclosed
CN-115385912-A Pyrazinopyrazinoquinolinone derivatives, preparation method and medical application thereof 浙江海正药业股份有限公司 2022-11-25 CN disclosed