SCHEMBL28565488

SCHEMBL28565488

COc1c[c]c(O)c(Cl)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 3/20 0.33
NPC1 O15118 2/20 0.33
MCL1 Q07820 2/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
RAB9A P51151 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
ABL1 P00519 1/20 0.31
ABCB1 P08183 1/20 0.31
BCR P11274 1/20 0.31
TP53 P04637 1/20 0.31
MAPK1 P28482 1/20 0.31
CASP3 P42574 1/20 0.31
SENP8 Q96LD8 1/20 0.31
SENP7 Q9BQF6 1/20 0.31
SENP6 Q9GZR1 1/20 0.31
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16056542 0.78 CYP3A4 (0.48) CYP3A4ALDH1A1MAPTNPC1MCL1
SCHEMBL2351365 0.78 ALDH1A1 (0.38) ALDH1A1NPC1CA1CA2GAA
SCHEMBL1638474 0.77 CYP3A4 (0.37) CYP3A4ALDH1A1MAPTNPC1MCL1
SCHEMBL27542323 0.77 ALDH1A1 (0.36) ALDH1A1CA1CA2
SCHEMBL2164186 0.77 CA12 (0.41) CYP3A4ALDH1A1MAPTCA1CA2
SCHEMBL2351389 0.75 ALDH1A1 (0.35) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL20397 0.72
SCHEMBL6912657 0.72 CA2 (0.57) CYP3A4ALDH1A1MAPTCA1CA2
SCHEMBL27743256 0.71 TAAR1 (0.33) ALDH1A1
SCHEMBL29025470 0.70 CYP3A4 (0.50) CYP3A4ALDH1A1MAPTNPC1MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113286792-B N-chromen-4-one containing derivatives for the treatment and prevention of hepatitis b virus infection 豪夫迈·罗氏有限公司 2023-12-05 CN disclosed
CN-112996566-B Chroman-4-one derivatives for the treatment and prevention of hepatitis B virus infection 豪夫迈·罗氏有限公司 2023-11-03 CN disclosed
CN-113286792-A N-containing chromen-4-one derivatives for the treatment and prevention of hepatitis B virus infection 豪夫迈·罗氏有限公司 2021-08-20 CN disclosed
CN-112996566-A Chroman-4-one derivatives for the treatment and prevention of hepatitis B virus infection 豪夫迈·罗氏有限公司 2021-06-18 CN disclosed
CN-112912371-A Flavone derivatives for treating and preventing hepatitis B virus diseases 豪夫迈·罗氏有限公司 2021-06-04 CN disclosed