SCHEMBL28569830

SCHEMBL28569830

CC(C)n1cc(C(N)=O)c(=O)c2cc(I)ccc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K2 P36507 3/20 0.37
MAP2K1 Q02750 3/20 0.37
KDM4E B2RXH2 2/20 0.37
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
MAP3K5 Q99683 2/20 0.34
CCNT1 O60563 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CDK9 P50750 1/20 0.34
GRM2 Q14416 1/20 0.34
PTPN1 P18031 1/20 0.33
DNMT1 P26358 1/20 0.33
PARP1 P09874 1/20 0.33
XDH P47989 1/20 0.33
CAPN1 P07384 1/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4154022 0.88 KDM4E (0.42) KDM4ECNR1CNR2MEN1KMT2A
SCHEMBL28564024 0.82 KDM4E (0.50) MAP2K2MAP2K1KDM4ECNR1CNR2
SCHEMBL3001658 0.81 LMNA (0.52) MAP2K2MAP2K1KDM4EMEN1KMT2A
SCHEMBL29594757 0.78 ALDH1A1 (0.53) MAP2K2MAP2K1KDM4ECNR1CNR2
SCHEMBL28450562 0.78 ALDH1A1 (0.53) MAP2K2MAP2K1KDM4ECNR1CNR2
SCHEMBL3004233 0.75 KDM4E (0.42) KDM4ECNR1CNR2PTPN1DNMT1
SCHEMBL4158355 0.75 KDM4E (0.44) MAP2K2MAP2K1KDM4ECNR1CNR2
SCHEMBL4141571 0.75 KDM4E (0.41) MAP2K2MAP2K1KDM4ECNR1CNR2
SCHEMBL28914037 0.75 MEN1 (0.60) MAP2K2MAP2K1KDM4ECNR1CNR2
SCHEMBL2990529 0.74 METTL3 (0.50) MAP2K2MAP2K1KDM4ECNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109942653-B Erythromycin derivative and preparation method thereof 北京理工大学 2021-06-25 CN disclosed
CN-109942654-B Macrolide and quinolone heterocomplex and preparation method thereof 北京理工大学 2021-06-11 CN disclosed