SCHEMBL28569853

SCHEMBL28569853

CN1CCC(Oc2c(O[C@H]3CCOC3)ccc(OC(N)=O)c2C#N)C(F)(F)C1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 12/20 0.36
PDE4A P27815 6/20 0.36
PDE4B Q07343 6/20 0.36
PDE4C Q08493 6/20 0.36
EGFR P00533 1/20 0.36
ERBB2 P04626 1/20 0.36
MAPK8 P45983 1/20 0.35
MAPK9 P45984 1/20 0.35
CHEK1 O14757 2/20 0.34
FASN P49327 3/20 0.33
FGFR4 P22455 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28569856 1.00 PDE4D (0.36) PDE4DPDE4APDE4BPDE4CEGFR
SCHEMBL21886669 0.87 EGFR (0.37) PDE4DPDE4APDE4BPDE4CEGFR
SCHEMBL28564240 0.87 EGFR (0.37) PDE4DPDE4APDE4BPDE4CEGFR
SCHEMBL28555129 0.85 ERBB2 (0.39) PDE4DPDE4APDE4BPDE4CEGFR
SCHEMBL21886628 0.85 ERBB2 (0.39) PDE4DPDE4APDE4BPDE4CEGFR
SCHEMBL21886730 0.82 CHEK1 (0.38) PDE4DPDE4APDE4BPDE4CEGFR
SCHEMBL30513784 0.82 CHEK1 (0.38) PDE4DPDE4APDE4BPDE4CEGFR
SCHEMBL28559957 0.82 CHEK1 (0.38) PDE4DPDE4APDE4BPDE4CEGFR
SCHEMBL21886635 0.80 EGFR (0.35) EGFRERBB2CHEK1
SCHEMBL30988767 0.75 GPR119 (0.37) PDE4DPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118255772-A Quinazoline derivatives as antitumor agents 苏州赞荣医药科技有限公司 2024-06-28 CN disclosed
CN-112654612-A Quinazoline derivatives as antitumor agents 苏州赞荣医药科技有限公司 2021-04-13 CN disclosed