SCHEMBL28572004

SCHEMBL28572004

O=C(/C=C/c1ccc2c(c1)OCCO2)NC(Cc1ccccc1)Cn1ccnc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.46
MAPT P10636 5/20 0.46
KDM4E B2RXH2 3/20 0.46
LMNA P02545 2/20 0.46
TP53 P04637 1/20 0.46
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 1/20 0.45
POLB P06746 1/20 0.45
KMT2A Q03164 1/20 0.45
ALOX15 P16050 1/20 0.44
TBXAS1 P24557 1/20 0.43
HDAC1 Q13547 1/20 0.41
HCAR2 Q8TDS4 1/20 0.41
PKM P14618 1/20 0.41
PLK1 P53350 1/20 0.41
TRPM8 Q7Z2W7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30566316 1.00 TRPV1 (0.46) TRPV1MAPTKDM4ELMNATP53
SCHEMBL28565823 0.86 MAPT (0.46) TRPV1MAPTKDM4ELMNATP53
SCHEMBL28571346 0.84 TBXAS1 (0.47) LMNAMEN1POLBKMT2ATBXAS1
SCHEMBL30566315 0.84 CYP19A1 (0.50) TRPV1MAPTKDM4ELMNATP53
SCHEMBL30566320 0.84 KDM4E (0.45) KDM4ESMN1; SMN2ALDH1A1ALOX15TBXAS1
SCHEMBL28566380 0.84 KDM4E (0.45) KDM4ESMN1; SMN2ALDH1A1ALOX15TBXAS1
SCHEMBL28571445 0.84 CYP19A1 (0.50) TRPV1MAPTKDM4ELMNATP53
SCHEMBL28433866 0.78 ALDH1A1 (0.51) LMNAALDH1A1MEN1KMT2ATBXAS1
SCHEMBL28433865 0.78 ALDH1A1 (0.51) LMNAALDH1A1MEN1KMT2ATBXAS1
SCHEMBL28569168 0.77 HDAC8 (0.45) MAPTKDM4ESMN1; SMN2ALDH1A1TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112142673-A Arylalkenole derivative and preparation method and application thereof 聊城大学 2020-12-29 CN claimed
CN-112142673-B Aryl alkene azole derivative and preparation method and application thereof 聊城大学 2023-06-30 CN disclosed
CN-112142673-A Arylalkenole derivative and preparation method and application thereof 聊城大学 2020-12-29 CN disclosed