SCHEMBL28573752

SCHEMBL28573752

CC(C)c1c(C(N)=O)ccc(C(F)(F)F)c1C(C)C

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.36
CTSK P43235 1/20 0.36
CES2 O00748 2/20 0.36
IRAK4 Q9NWZ3 1/20 0.34
MAPK10 P53779 2/20 0.33
PARP1 P09874 2/20 0.33
DGAT1 O75907 1/20 0.33
LMNA P02545 2/20 0.32
XBP1 P17861 1/20 0.32
GPR52 Q9Y2T5 2/20 0.32
GAA P10253 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
AKT1 P31749 1/20 0.31
CDC7 O00311 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2882576 0.83 IRAK4 (0.44) IRAK4PARP1DGAT1MEN1ALDH1A1
SCHEMBL28386490 0.77 DGAT1 (0.43) CES2IRAK4PARP1DGAT1GAA
SCHEMBL27721639 0.76 KCNK3 (0.39) CTSSCTSKIRAK4AKT1
SCHEMBL25557189 0.75 CES2 (0.42) CES2GAAALDH1A1AKT1
SCHEMBL5461078 0.75 CES2 (0.42) CES2GPR52GAAALDH1A1AKT1
SCHEMBL28887386 0.74 SIRT3 (0.40) IRAK4PARP1DGAT1LMNAALDH1A1
SCHEMBL8011592 0.74 IRAK4 (0.38) IRAK4DGAT1ALDH1A1MAPTKMT2A
SCHEMBL5182718 0.73 TAS2R14 (0.40) CTSSCES2MAPK10PARP1DGAT1
SCHEMBL6599789 0.73 ERN1 (0.43) IRAK4DGAT1ALDH1A1MAPTKMT2A
SCHEMBL28882111 0.73 IRAK4 (0.37) IRAK4PARP1DGAT1MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112794831-B 3- (3' -hydroxybutyl) isobenzofuran-1 (3H) -one derivative, composition, preparation method and application thereof 北京理工大学 2021-07-27 CN disclosed
CN-112794831-A 3- (3' -hydroxybutyl) isobenzofuran-1 (3H) -one derivative, composition, preparation method and application thereof 北京理工大学 2021-05-14 CN disclosed