SCHEMBL28575489

SCHEMBL28575489

CCOC(=O)c1nc(-c2ccccc2)[nH]c1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.49
PIN1 Q13526 5/20 0.49
HSD17B10 Q99714 3/20 0.47
MAPK1 P28482 2/20 0.47
USP2 O75604 1/20 0.47
TSHR P16473 1/20 0.47
TARBP2 Q15633 1/20 0.47
ROCK2 O75116 1/20 0.46
KDM4E B2RXH2 4/20 0.46
ALDH1A1 P00352 3/20 0.46
HPGD P15428 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
RAB9A P51151 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TRPM8 Q7Z2W7 1/20 0.46
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27475261 0.82 PIN1 (0.68) PIN1HSD17B10MAPK1USP2TSHR
SCHEMBL7989950 0.82 MAPK13 (0.51) DGAT1PIN1HSD17B10TARBP2KDM4E
SCHEMBL28582964 0.81 TARBP2 (0.54) PIN1HSD17B10MAPK1USP2TSHR
SCHEMBL6520020 0.80 PIN1 (0.52) PIN1HSD17B10MAPK1USP2TSHR
SCHEMBL21374324 0.80 PIN1 (0.52) PIN1HSD17B10MAPK1USP2TSHR
SCHEMBL15592594 0.80 HSD17B10 (0.56) PIN1HSD17B10MAPK1USP2TSHR
SCHEMBL31110150 0.78 PIN1 (0.50) DGAT1PIN1MAPK1HPGDERCC1
SCHEMBL17790243 0.78 KDM4E (0.40) HSD17B10KDM4EALDH1A1HPGDMAPT
SCHEMBL9049053 0.77 KDM4E (0.50) HSD17B10TSHRTARBP2KDM4EALDH1A1
SCHEMBL17803252 0.77 KDM4E (0.58) PIN1HSD17B10KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112759551-B 2, 5-substituent 1H-imidazole-4-carboxylate compound and synthetic purification method thereof 宝鸡文理学院 2023-10-27 CN disclosed
CN-112759551-A 2, 5-substituent 1H-imidazole-4-carboxylic ester compound and synthesis and purification method thereof 宝鸡文理学院 2021-05-07 CN disclosed