SCHEMBL2857574

SCHEMBL2857574

O=C(Nc1ccccc1C(F)(F)F)Oc1cnn(-c2ccccc2)c1C(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.50
POLB P06746 3/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
KDM4E B2RXH2 4/20 0.48
ALDH1A1 P00352 2/20 0.48
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
NR3C1 P04150 1/20 0.44
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
KCNJ6 P48051 1/20 0.43
KCNJ5 P48544 1/20 0.43
KCNJ3 P48549 1/20 0.43
EPHB3 P54753 1/20 0.42
MET P08581 1/20 0.41
AXL P30530 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854596 0.91 TP53 (0.46) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2850871 0.89 NPC1 (0.51) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2856355 0.88 RAB9A (0.52) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2860786 0.88 MAPT (0.49) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2850763 0.87 MAPT (0.48) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2850725 0.86 MAPT (0.54) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2850610 0.84 MAPT (0.40) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2853256 0.84 SMN1; SMN2 (0.46) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2853459 0.83 MAPT (0.52) MAPTPOLBKDM4EALDH1A1CYP1A2
SCHEMBL2853255 0.82 HSP90AA1 (0.48) MAPTPOLBSMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed