SCHEMBL2854596

SCHEMBL2854596

O=C(Nc1ccccc1C(F)(F)F)Oc1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.46
GAA P10253 2/20 0.46
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
NR3C1 P04150 1/20 0.41
MAPT P10636 4/20 0.41
POLB P06746 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GRIK1 P39086 1/20 0.41
KMT2A Q03164 2/20 0.41
CCR1 P32246 2/20 0.40
EPHB3 P54753 1/20 0.40
MEN1 O00255 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850610 0.93 MAPT (0.40) TP53GAAKDM4EALDH1A1NR3C1
SCHEMBL2857574 0.91 MAPT (0.50) KDM4EALDH1A1NR3C1MAPTPOLB
SCHEMBL2857353 0.91 CCR1 (0.47) TP53GAAKDM4EALDH1A1MAPT
SCHEMBL2852552 0.91 MEN1 (0.51) KDM4EALDH1A1MAPTPOLBSMN1; SMN2
SCHEMBL2848541 0.90 RAB9A (0.43) KDM4EALDH1A1MAPTPOLBSMN1; SMN2
SCHEMBL2859508 0.89 CYP1A2 (0.46) KDM4EALDH1A1MAPTPOLBSMN1; SMN2
SCHEMBL2855775 0.88 P2RY1 (0.44) TP53GAAKDM4EALDH1A1NR3C1
SCHEMBL2852820 0.87 TMPRSS4 (0.45) TP53ALDH1A1MAPTCCR1HTT
SCHEMBL2857074 0.86 LPAR1 (0.42) KDM4EALDH1A1MAPTPOLBSMN1; SMN2
SCHEMBL2858110 0.86 KDM4E (0.44) GAAKDM4EALDH1A1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed