SCHEMBL28577700

SCHEMBL28577700

Cc1cc(C=O)ccc1NC(=O)C(C)(C)C.Cc1ccccc1NC(=O)C(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.50
PDK2 Q15119 1/20 0.50
PDK3 Q15120 1/20 0.50
PDK4 Q16654 1/20 0.50
CETP P11597 1/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
HPGD P15428 2/20 0.45
ALDH1A1 P00352 1/20 0.45
MMP1 P03956 4/20 0.44
MMP2 P08253 4/20 0.44
MMP9 P14780 4/20 0.44
EGFR P00533 1/20 0.43
NPSR1 Q6W5P4 3/20 0.43
PKM P14618 1/20 0.43
DDX3X O00571 1/20 0.42
MAPT P10636 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 1/20 0.42
STAT1 P42224 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28572812 0.93 TP53 (0.44) PDK1PDK2PDK3PDK4CETP
SCHEMBL397003 0.83 PDK1 (0.67) PDK1PDK2PDK3PDK4CETP
SCHEMBL15332043 0.78 CETP (0.47) CETPRAB9AHPGDALDH1A1MMP1
SCHEMBL7069760 0.77 POLB (0.44) NPC1RAB9AHPGDALDH1A1MMP1
SCHEMBL7013927 0.76 ALDH1A1 (0.52) NPC1RAB9AHPGDALDH1A1NPSR1
SCHEMBL19448892 0.75 CETP (0.49) PDK1PDK2PDK3PDK4CETP
SCHEMBL5164739 0.74 SMN1; SMN2 (0.44) NPC1RAB9AHPGDALDH1A1NPSR1
SCHEMBL5706504 0.73 CETP (0.71) PDK1PDK2PDK3PDK4CETP
SCHEMBL15427825 0.72 CETP (0.57) PDK1PDK2PDK3PDK4CETP
SCHEMBL6349201 0.72 PDK1 (0.70) PDK1PDK2PDK3PDK4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113024399-A Pharmaceutical intermediate compound and preparation method and application thereof 华东理工大学 2021-06-25 CN claimed
CN-113024399-B Pharmaceutical intermediate compound and preparation method and application thereof 华东理工大学 2022-09-09 CN disclosed
CN-113024469-A Synthesis method of telmisartan intermediate 华东理工大学 2021-06-25 CN disclosed
CN-113024399-A Pharmaceutical intermediate compound and preparation method and application thereof 华东理工大学 2021-06-25 CN disclosed