SCHEMBL2858036

SCHEMBL2858036

CC(C)(C)OC(=O)NC(=N)c1cccc(NC(=O)c2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.44
MAPT P10636 3/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
TP53 P04637 1/20 0.42
THRB P10828 1/20 0.42
NR1H4 Q96RI1 1/20 0.42
MALT1 Q9UDY8 9/20 0.42
LMNA P02545 1/20 0.42
ATM Q13315 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4882354 0.88 NPC1 (0.49) BRAFMAPTNPC1RAB9ANR1H4
SCHEMBL2850892 0.82 NR1H4 (0.53) BRAFMAPTNPC1RAB9ANR1H4
SCHEMBL2858034 0.81 BRAF (0.43) BRAFMAPTTP53THRBNR1H4
SCHEMBL14539344 0.81 KDM4E (0.52) BRAFMAPTNR1H4MALT1KDM4E
SCHEMBL2853811 0.80 SMN1; SMN2 (0.60) BRAFMAPTNPC1RAB9ATP53
SCHEMBL2852818 0.80 NPC1 (0.50) BRAFMAPTNPC1RAB9ATP53
SCHEMBL14539343 0.79 NR1H4 (0.47) BRAFMAPTNR1H4MALT1KDM4E
SCHEMBL13513708 0.78 KDM4E (0.53) BRAFMAPTMALT1KDM4EALDH1A1
SCHEMBL2852028 0.77 MAPT (0.46) BRAFMAPTTP53THRBNR1H4
SCHEMBL2857034 0.77 KDM4E (0.62) BRAFMAPTNPC1RAB9ANR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed