SCHEMBL28581983

SCHEMBL28581983

CC(CCC(NC(=O)c1nccn1C)C(N)=O)=C(C)C(N)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.40
NAMPT P43490 1/20 0.39
TGM2 P21980 1/20 0.35
LMNA P02545 2/20 0.34
KMT2A Q03164 2/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
CNR1 P21554 2/20 0.33
CNR2 P34972 2/20 0.33
HPGDS O60760 1/20 0.32
POLB P06746 1/20 0.32
F2 P00734 1/20 0.32
PRSS1 P07477 1/20 0.32
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA9 Q16790 1/20 0.31
FDPS P14324 1/20 0.31
ROCK2 O75116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31028374 0.87 SMYD3 (0.42) SMYD3NAMPTTGM2LMNAKMT2A
SCHEMBL28596375 0.79 P2RX7 (0.41) KMT2ACNR1CNR2HPGDSCA12
SCHEMBL28598466 0.77 TGM2 (0.35) TGM2HPGDSCA12CA1CA9
SCHEMBL28584273 0.75 GRM5 (0.36) HPGDSCA12CA1CA9
SCHEMBL8338299 0.72 SMYD3 (0.47) SMYD3CNR1CNR2HPGDS
SCHEMBL28586865 0.71 ACACB (0.38) HPGDSCA12CA1CA9
SCHEMBL106846 0.69 NAMPT (0.53) SMYD3NAMPTLMNAKMT2AALDH1A1
SCHEMBL2363843 0.67 SMYD3 (0.49) SMYD3NAMPTLMNAKMT2AALDH1A1
SCHEMBL28593255 0.64 NOD1 (0.34)
SCHEMBL10099637 0.64 NAMPT (0.54) SMYD3NAMPTLMNAKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112789040-A Transglutaminase 2(TG2) inhibitors 思达利医药公司 2021-05-11 CN claimed
CN-112789040-A Transglutaminase 2(TG2) inhibitors 思达利医药公司 2021-05-11 CN disclosed