SCHEMBL8338299

SCHEMBL8338299

Cn1ccnc1C(=O)N[C@@H](CC1CCCCC1)C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.47
CNR2 P34972 11/20 0.44
CNR1 P21554 1/20 0.44
MAPK11 Q15759 4/20 0.43
MAPK14 Q16539 4/20 0.43
HPGDS O60760 1/20 0.41
HTRA1 Q92743 1/20 0.40
GRN P28799 1/20 0.40
SORT1 Q99523 1/20 0.40
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP3 P08254 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8336645 0.77 MAPK11 (0.47) CNR2CNR1MAPK11MAPK14HPGDS
SCHEMBL8339904 0.75 MAPK11 (0.45) CNR2CNR1MAPK11MAPK14HPGDS
SCHEMBL31028374 0.75 SMYD3 (0.42) SMYD3CNR2CNR1HPGDS
SCHEMBL8334677 0.74 LONP1 (0.63) CNR2CNR1
SCHEMBL8339907 0.74 CNR2 (0.54) CNR2CNR1MAPK11MAPK14
SCHEMBL8337500 0.74 CTSK (0.53) CNR2CNR1MAPK11MAPK14HPGDS
SCHEMBL8337771 0.72 CTSK (0.51) CNR2CNR1MAPK11MAPK14HPGDS
SCHEMBL28581983 0.72 SMYD3 (0.40) SMYD3CNR2CNR1HPGDS
SCHEMBL21162958 0.71 F2RL1 (0.68)
SCHEMBL21162774 0.71 F2RL1 (0.68)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004017911-A2 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2004-03-04 WO disclosed