SCHEMBL28583221

SCHEMBL28583221

c1c[nH]c(N2CCCNC2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 6/20 0.38
CHRNA4 P43681 6/20 0.38
HTR1A P08908 6/20 0.35
HTR3A P46098 6/20 0.35
HTR7 P34969 5/20 0.35
HTR2B P41595 5/20 0.35
HTR6 P50406 5/20 0.35
USP2 O75604 2/20 0.33
ALDH1A1 P00352 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
CXCR4 P61073 2/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
GFER P55789 1/20 0.31
CYP1A2 P05177 1/20 0.31
HTR1D P28221 4/20 0.31
HTR2A P28223 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28106504 0.80
SCHEMBL261863 0.80 GFER (0.39) USP2ALDH1A1TSHRNPC1RAB9A
Piperazine SCHEMBL28080108 0.79 USP2 (0.38) CHRNB2CHRNA4HTR1AHTR3AHTR7
SCHEMBL1478216 0.78 NPC1 (0.41) USP2ALDH1A1TSHRNPC1RAB9A
SCHEMBL4491073 0.76 ADRB1 (0.48) HTR1AHTR3AHTR7HTR2BHTR6
SCHEMBL28697522 0.73 ADRB1 (0.32) HTR1AHTR6HTR2AHTR2C
SCHEMBL2051022 0.71 HTR3A (0.57) CHRNB2CHRNA4HTR1AHTR3AHTR7
SCHEMBL7189439 0.69 HDAC8 (0.34)
SCHEMBL3833537 0.68 LMNA (0.48) USP2ALDH1A1TSHRNPC1RAB9A
SCHEMBL21047844 0.68 NPC1 (0.33) NPC1RAB9AGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071532-B FGFR4 inhibitor, preparation method and application thereof 江苏豪森药业集团有限公司 2021-04-27 CN disclosed