SCHEMBL28583306

SCHEMBL28583306

CCC(=O)Nc1ccc(Nc2nc(-c3ccc(C)cc3)cs2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.69
RAB9A P51151 2/20 0.69
SMN1; SMN2 Q16637 2/20 0.69
MAPT P10636 6/20 0.67
GAA P10253 4/20 0.67
AMY1A P0DUB6 2/20 0.67
ALOX5 P09917 2/20 0.67
MEN1 O00255 3/20 0.62
KMT2A Q03164 3/20 0.62
PTGS2 P35354 1/20 0.60
NAMPT P43490 1/20 0.59
ALDH1A1 P00352 2/20 0.56
TDP1 Q9NUW8 2/20 0.56
USP2 O75604 1/20 0.56
LMNA P02545 1/20 0.56
THRB P10828 1/20 0.56
HPGD P15428 1/20 0.56
ALOX15 P16050 1/20 0.56
TSHR P16473 1/20 0.56
ALOX12 P18054 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28575173 0.89 MAPT (0.66) NPC1RAB9ASMN1; SMN2MAPTGAA
SCHEMBL28575151 0.89 ALOX5 (0.69) NPC1RAB9ASMN1; SMN2MAPTGAA
SCHEMBL28575303 0.89 MAPT (0.66) NPC1RAB9ASMN1; SMN2MAPTGAA
SCHEMBL28594556 0.89 CSNK2A1 (0.67) NPC1RAB9ASMN1; SMN2MAPTGAA
SCHEMBL14085825 0.87 HDAC1 (0.67) NPC1RAB9ASMN1; SMN2MAPTGAA
SCHEMBL28575126 0.86 ALOX5 (0.64) NPC1RAB9ASMN1; SMN2MAPTGAA
SCHEMBL28575125 0.86 MAPT (0.72) NPC1RAB9ASMN1; SMN2MAPTGAA
SCHEMBL17320209 0.84 ALOX5 (0.85) NPC1RAB9ASMN1; SMN2MAPTGAA
SCHEMBL28583387 0.84 ALOX5 (0.67) NPC1RAB9ASMN1; SMN2MAPTGAA
SCHEMBL28579111 0.84 MAPT (0.59) NPC1RAB9ASMN1; SMN2MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113004219-A Thiazole ring-containing amide compound and preparation method and application thereof 贵州大学 2021-06-22 CN disclosed