SCHEMBL28586335

SCHEMBL28586335

C1CNCCNC1.O=S(=O)(Cl)c1cccc2cnccc12

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCZ Q05513 8/20 0.62
PRKD3 O94806 7/20 0.62
PRKCG P05129 7/20 0.62
PRKCB P05771 7/20 0.62
PRKCA P17252 7/20 0.62
PRKCH P24723 7/20 0.62
PRKCI P41743 7/20 0.62
PRKCE Q02156 7/20 0.62
PRKCQ Q04759 7/20 0.62
PRKCD Q05655 7/20 0.62
PRKD1 Q15139 7/20 0.62
ROCK2 O75116 7/20 0.62
CYP3A4 P08684 6/20 0.62
ROCK1 Q13464 6/20 0.62
PRKACA P17612 5/20 0.62
PRKACG P22612 5/20 0.62
PRKACB P22694 5/20 0.62
CYP2D6 P10635 5/20 0.62
SMN1; SMN2 Q16637 4/20 0.62
MEN1 O00255 4/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL115053 0.87 CYP3A4 (0.56) PRKCZPRKD3PRKCGPRKCBPRKCA
SCHEMBL29546384 0.87 CYP3A4 (0.56) PRKCZPRKD3PRKCGPRKCBPRKCA
Hydrochloric Acid SCHEMBL987360 0.85 LMNA (0.57) PRKCZPRKD3PRKCGPRKCBPRKCA
Hydrochloric Acid SCHEMBL29469852 0.85 LMNA (0.57) PRKCZPRKD3PRKCGPRKCBPRKCA
Fasudil SCHEMBL6269832 0.77 ROCK2 (1.00) PRKCZPRKD3PRKCGPRKCBPRKCA
Fasudil SCHEMBL29381868 0.77 ROCK2 (1.00) PRKCZPRKD3PRKCGPRKCBPRKCA
Fasudil SCHEMBL4674 0.77 ROCK2 (1.00) PRKCZPRKD3PRKCGPRKCBPRKCA
Fasudil SCHEMBL29362990 0.77 ROCK2 (1.00) PRKCZPRKD3PRKCGPRKCBPRKCA
SCHEMBL28592488 0.77 PRKD3 (0.49) PRKCZPRKD3PRKCGPRKCBPRKCA
Fasudil SCHEMBL678615 0.76 ROCK2 (0.98) PRKCZPRKD3PRKCGPRKCBPRKCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112986409-A Method for detecting isoquinoline sulfonate genotoxic impurities in fasudil 南京亿华药业有限公司 2021-06-18 CN disclosed