SCHEMBL28587780

SCHEMBL28587780

N#Cc1cccc(COc2ccccc2-c2nc(C(=O)O)cc(=O)[nH]2)c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SGMS2 Q8NHU3 1/20 0.44
MRGPRX4 Q96LA9 4/20 0.44
FFAR1 O14842 1/20 0.43
FFAR4 Q5NUL3 1/20 0.43
PPIA P62937 1/20 0.43
PTGER1 P34995 2/20 0.42
ALKBH1 Q13686 1/20 0.41
PDE5A O76074 1/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
GRM5 P41594 1/20 0.41
XDH P47989 1/20 0.41
BRS3 P32247 1/20 0.41
SRD5A2 P31213 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28587829 0.89 SGMS2 (0.44) SGMS2MRGPRX4FFAR1FFAR4PPIA
SCHEMBL28587775 0.84 FFAR1 (0.53) FFAR1FFAR4ALKBH1XDH
SCHEMBL28583440 0.79 XDH (0.59) SGMS2MRGPRX4FFAR1FFAR4PPIA
SCHEMBL28587005 0.76 XDH (0.56) SGMS2MRGPRX4FFAR1FFAR4PPIA
SCHEMBL28568681 0.75 PDE5A (0.38) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL28593875 0.74 PDE5A (0.37) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL28587828 0.73 FFAR1 (0.52) MRGPRX4FFAR1FFAR4ALKBH1
SCHEMBL28593877 0.73 PDE5A (0.39) PTGER1PDE5APDE4APDE4BPDE4C
SCHEMBL28916533 0.72 XDH (0.53) SGMS2MRGPRX4FFAR1FFAR4PPIA
SCHEMBL13851581 0.69 POLB (0.63) PDE5APDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112979559-A 2-phenyl pyrimidine formic acid derivative and preparation method and application thereof 沈阳药科大学 2021-06-18 CN claimed
CN-112979559-A 2-phenyl pyrimidine formic acid derivative and preparation method and application thereof 沈阳药科大学 2021-06-18 CN disclosed