SCHEMBL28587775

SCHEMBL28587775

N#Cc1cccc(COc2ccc(-c3nc(C(=O)O)cc(=O)[nH]3)cc2)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 2/20 0.53
FFAR4 Q5NUL3 1/20 0.53
ALOX5 P09917 1/20 0.50
ALOX5AP P20292 1/20 0.50
ALKBH1 Q13686 1/20 0.49
DHODH Q02127 2/20 0.48
MCL1 Q07820 2/20 0.47
ADAMTS4 O75173 1/20 0.46
MMP13 P45452 1/20 0.46
MAOB P27338 2/20 0.46
XDH P47989 1/20 0.45
CYP19A1 P11511 1/20 0.45
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
KCNH2 Q12809 1/20 0.45
PRMT5 O14744 2/20 0.45
TDP2 O95551 1/20 0.44
CHEK2 O96017 1/20 0.44
MAOA P21397 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28587828 0.89 FFAR1 (0.52) FFAR1FFAR4ALOX5ALOX5APALKBH1
SCHEMBL28587780 0.84 SGMS2 (0.44) FFAR1FFAR4ALKBH1XDH
SCHEMBL28583439 0.78 XDH (0.61) FFAR1FFAR4ALOX5ALOX5APALKBH1
SCHEMBL28587004 0.75 ALKBH1 (0.64) FFAR1FFAR4ALOX5ALOX5APALKBH1
SCHEMBL28580883 0.74 PDE2A (0.44) XDH
SCHEMBL28593871 0.73 PDE2A (0.38) XDHCHEK2
SCHEMBL28587829 0.73 SGMS2 (0.44) FFAR1FFAR4ALKBH1DHODHXDH
SCHEMBL1247999 0.73 MAOB (0.63) FFAR1FFAR4ALOX5ALOX5APADAMTS4
SCHEMBL851377 0.72 MEN1 (0.68) FFAR1FFAR4ALKBH1MAOB
SCHEMBL18035933 0.72 PDE2A (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112979559-A 2-phenyl pyrimidine formic acid derivative and preparation method and application thereof 沈阳药科大学 2021-06-18 CN claimed
CN-112979559-A 2-phenyl pyrimidine formic acid derivative and preparation method and application thereof 沈阳药科大学 2021-06-18 CN disclosed