SCHEMBL2859008

SCHEMBL2859008

O=C(NCc1cccc(C(F)(F)F)c1)c1cnn(-c2cc(Cl)ccc2Cl)c1C(F)(F)F

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.66
HPGD P15428 1/20 0.66
CCR1 P32246 14/20 0.65
MEN1 O00255 1/20 0.53
PLA2G1B P04054 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
GAA P10253 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C19 P33261 1/20 0.53
KMT2A Q03164 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
ATG4B Q9Y4P1 1/20 0.53
HSP90AA1 P07900 2/20 0.50
MAPT P10636 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
HSP90AB1 P08238 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2857075 0.91 P2RX1 (0.57) LMNAHPGDCCR1HSP90AA1MAPT
SCHEMBL2859858 0.90 CCR1 (0.52) LMNAHPGDCCR1CYP1A2CYP3A4
SCHEMBL2850536 0.88 CCR1 (0.52) LMNAHPGDCCR1
SCHEMBL2859933 0.87 CCR1 (0.80) LMNAHPGDCCR1MEN1PLA2G1B
SCHEMBL2854432 0.87 CCR1 (0.68) LMNAHPGDCCR1MEN1PLA2G1B
SCHEMBL2852539 0.84 LMNA (0.52) LMNAHPGDCCR1MEN1PLA2G1B
SCHEMBL2856467 0.83 P2RX7 (0.51) LMNAHPGDCCR1HSP90AA1MAPT
SCHEMBL2860195 0.82 CCR1 (0.70) LMNAHPGDCCR1NPSR1
SCHEMBL2859642 0.82 CCR1 (0.73) HPGDCCR1MAPT
SCHEMBL2855376 0.81 CCR1 (0.60) LMNAHPGDCCR1MEN1PLA2G1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed