SCHEMBL2859083

SCHEMBL2859083

Cc1cccc(C(=O)C#CC(=O)NC2CCN(c3nc(C)cs3)C2)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 4/20 0.40
CDK2 P24941 4/20 0.40
CYP2C19 P33261 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CTDSP1 Q9GZU7 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ALDH1A1 P00352 1/20 0.37
SMPD3 Q9NY59 1/20 0.36
LMNA P02545 1/20 0.36
BTK Q06187 1/20 0.36
CCR2 P41597 2/20 0.36
POLB P06746 1/20 0.36
MAPK1 P28482 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2858190 0.91 MEN1 (0.38) CCNE1CDK2CYP2C19SMN1; SMN2NPC1
SCHEMBL2854222 0.89 SMN1; SMN2 (0.40) CCNE1CDK2CYP2C19SMN1; SMN2NPC1
SCHEMBL2858043 0.87 CCNE1 (0.40) CCNE1CDK2CYP2C19SMN1; SMN2NPC1
SCHEMBL973019 0.86 BTK (0.38) CCNE1CDK2SMPD3BTKHRH3
SCHEMBL2862996 0.83 CCNE1 (0.38) CCNE1CDK2CYP2C19SMN1; SMN2NPC1
SCHEMBL2855060 0.83 ALDH1A1 (0.43) SMN1; SMN2MEN1KMT2AALDH1A1SMPD3
SCHEMBL2853786 0.80 LMNA (0.38) CYP2C19SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL4698213 0.80 DRD2 (0.40) CCNE1CDK2SMN1; SMN2NPC1RAB9A
SCHEMBL973545 0.80 BTK (0.45) SMPD3BTKHRH3
SCHEMBL974804 0.80 SMN1; SMN2 (0.41) CYP2C19SMN1; SMN2NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968957-B1 SUBSTITUTED THIAZOLES AND THEIR USE FOR PRODUCING DRUGS GRUENENTHAL GMBH (DE) 2010-01-20 EP claimed