SCHEMBL2862996

SCHEMBL2862996

Cc1cccc(C(=O)C#CC(=O)NC2CCN(c3ncc(C)s3)C2)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 4/20 0.38
CDK2 P24941 4/20 0.38
BTK Q06187 1/20 0.38
CYP2C19 P33261 1/20 0.37
CTDSP1 Q9GZU7 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 1/20 0.37
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
CHRNA7 P36544 2/20 0.36
CCR2 P41597 2/20 0.36
MAPK1 P28482 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ACKR3 P25106 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2856320 0.89 CHRNA7 (0.40) CCNE1CDK2BTKKMT2ACHRNA7
SCHEMBL975864 0.86 BTK (0.38) BTKCHRNA7HRH3ACKR3
SCHEMBL2858043 0.85 CCNE1 (0.40) CCNE1CDK2BTKCYP2C19CTDSP1
SCHEMBL2859083 0.83 CCNE1 (0.40) CCNE1CDK2BTKCYP2C19CTDSP1
SCHEMBL2856121 0.83 PAK1 (0.40) BTKMEN1KMT2AALDH1A1CHRNA7
SCHEMBL2858190 0.80 MEN1 (0.38) CCNE1CDK2BTKCYP2C19CTDSP1
SCHEMBL973764 0.80 BTK (0.45) BTKCHRNA7HRH3ACKR3
SCHEMBL974821 0.80 HRH3 (0.38) BTKCHRNA7HRH3ACKR3
SCHEMBL974009 0.79 RAB9A (0.39) CCNE1CDK2BTKRAB9AHRH3
SCHEMBL971211 0.79 CHRM5 (0.41) BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968957-B1 SUBSTITUTED THIAZOLES AND THEIR USE FOR PRODUCING DRUGS GRUENENTHAL GMBH (DE) 2010-01-20 EP claimed