SCHEMBL2859419

SCHEMBL2859419

O=C(NC(c1cccnc1)c1cccnc1)Oc1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.45
POLB P06746 2/20 0.38
MAPT P10636 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
HTT P42858 1/20 0.37
CCR1 P32246 2/20 0.36
ACHE P22303 1/20 0.36
ABCB1 P08183 1/20 0.36
NR3C1 P04150 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2853091 0.83 MAPT (0.49) CYP3A4POLBMAPTSMN1; SMN2CCR1
SCHEMBL2858436 0.83 MEN1 (0.46) CYP3A4MAPTSMN1; SMN2HTTKDM4E
SCHEMBL2862815 0.83 DRD2 (0.41) CYP3A4POLBMAPTSMN1; SMN2CCR1
SCHEMBL2854457 0.82 CYP3A4 (0.43) CYP3A4POLBMAPTSMN1; SMN2HTT
SCHEMBL2854852 0.81 ABCB1 (0.49) SMN1; SMN2HTTCCR1ABCB1KDM4E
SCHEMBL2853193 0.79 MAPT (0.43) MAPTSMN1; SMN2CCR1ABCB1
SCHEMBL2857729 0.78 CNR1 (0.53) MAPTKDM4E
SCHEMBL2850524 0.78 MAPT (0.43) CYP3A4MAPTSMN1; SMN2ACHENR3C1
SCHEMBL2860795 0.77 KMT2A (0.46) CYP3A4POLBMAPTSMN1; SMN2ACHE
SCHEMBL2852244 0.77 MAPT (0.48) POLBMAPTSMN1; SMN2ACHENR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed