SCHEMBL2862815

SCHEMBL2862815

O=C(NC(c1ccccn1)c1ccccn1)Oc1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.41
MAPT P10636 3/20 0.38
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
MALT1 Q9UDY8 2/20 0.37
CCR1 P32246 3/20 0.36
MAPK1 P28482 2/20 0.36
ACHE P22303 1/20 0.36
CNR1 P21554 2/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2859870 0.89 TLR7 (0.38) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2854514 0.87 CNR2 (0.35) DRD2MAPTPOLBSMN1; SMN2KDM4E
SCHEMBL2860499 0.86 RAB9A (0.35) DRD2MAPTPOLBSMN1; SMN2KDM4E
SCHEMBL2856129 0.85 DRD2 (0.35) DRD2MAPTMALT1MAPK1CNR1
SCHEMBL2860428 0.83 KDM4E (0.52) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2859419 0.83 CYP3A4 (0.45) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2858119 0.82 MAPT (0.43) DRD2MAPTPOLBSMN1; SMN2KDM4E
SCHEMBL2854676 0.81 ALDH1A1 (0.45) MAPTSMN1; SMN2KDM4EALDH1A1MALT1
SCHEMBL2848353 0.79 SMN1; SMN2 (0.48) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2848317 0.79 MAPT (0.46) MAPTPOLBSMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed