SCHEMBL28596019

SCHEMBL28596019

CN1CCC(n2c(=O)[nH]c3cc(B4OC(C)(C)C(C)(C)O4)ccc32)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.47
DRD2 P14416 2/20 0.47
HTR2A P28223 2/20 0.47
DRD3 P35462 2/20 0.47
ADRA2A P08913 1/20 0.47
SLC6A4 P31645 1/20 0.47
SIRT2 Q8IXJ6 1/20 0.46
PLD1 Q13393 1/20 0.44
CHRM1 P11229 4/20 0.42
CHRM2 P08172 3/20 0.42
CHRM4 P08173 3/20 0.42
CHRM3 P20309 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
BACE1 P56817 1/20 0.42
OPRM1 P35372 3/20 0.41
TNKS O95271 1/20 0.41
TNKS2 Q9H2K2 1/20 0.41
KCNH2 Q12809 2/20 0.40
CHRM5 P08912 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22191144 0.83 PGR (0.51) SIRT2CHRM1CHRM2CHRM4CHRM3
SCHEMBL22191190 0.82 CHRM1 (0.46) SIRT2CHRM1CHRM2CHRM4CHRM3
SCHEMBL14250830 0.78 LMNA (0.45) BACE1
SCHEMBL13823764 0.77 OPRM1 (0.61) HTR1ADRD2HTR2ADRD3ADRA2A
SCHEMBL28604447 0.76 OPRM1 (0.60) HTR1ADRD2HTR2ADRD3ADRA2A
SCHEMBL10316252 0.76 DRD2 (0.76) HTR1ADRD2HTR2ADRD3ADRA2A
SCHEMBL18198763 0.74 CA1 (0.38) BACE1
SCHEMBL5004813 0.74 BACE1 (0.33) HTR1ADRD2HTR2ADRD3ADRA2A
SCHEMBL14515170 0.73 OPRM1 (0.60) HTR1ADRD2HTR2ADRD3ADRA2A
SCHEMBL4152396 0.73 CYP2D6 (0.70) DRD2PLD1CHRM1CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113166139-A Pyrrolo [2,3-b ] pyridines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-07-23 CN disclosed