SCHEMBL28596233

SCHEMBL28596233

COc1ccc(N)c(C(=O)OC(=O)c2ccccc2N)c1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.51
HSD17B10 Q99714 9/20 0.51
CFTR P13569 1/20 0.51
TSHR P16473 4/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
KDM4E B2RXH2 4/20 0.42
HPGD P15428 3/20 0.42
RCE1 Q9Y256 1/20 0.42
POLB P06746 2/20 0.39
TDP1 Q9NUW8 3/20 0.39
ADRA2B P18089 1/20 0.39
PTGS1 P23219 1/20 0.39
IDO1 P14902 1/20 0.38
MAPT P10636 1/20 0.38
CTSD P07339 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
GLA P06280 2/20 0.38
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29501303 0.88 TUBB1 (0.44) ALDH1A1TSHRSMN1; SMN2KDM4EPOLB
SCHEMBL28596231 0.88 TUBB1 (0.44) ALDH1A1TSHRSMN1; SMN2KDM4EPOLB
SCHEMBL28415491 0.79 KDM4E (0.47) ALDH1A1HSD17B10CFTRTSHRSMN1; SMN2
SCHEMBL28701486 0.78 CTSD (0.47) ALDH1A1HSD17B10CFTRTSHRSMN1; SMN2
SCHEMBL2367627 0.76 ALDH1A1 (0.69) ALDH1A1HSD17B10CFTRTSHRSMN1; SMN2
SCHEMBL27422765 0.75 ALDH1A1 (0.67) ALDH1A1HSD17B10CFTRTSHRSMN1; SMN2
SCHEMBL339501 0.74 TUBB1 (0.45) ALDH1A1TSHRSMN1; SMN2TDP1IDO1
SCHEMBL29501305 0.74 L3MBTL1 (0.49) ALDH1A1TSHRSMN1; SMN2KDM4EPOLB
SCHEMBL1321669 0.74 MAPT (0.51) ALDH1A1HSD17B10TSHRSMN1; SMN2KDM4E
SCHEMBL348929 0.74 L3MBTL1 (0.49) ALDH1A1TSHRSMN1; SMN2KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113121427-B Quinoline derivative and preparation method and application thereof 广东工业大学 2022-04-01 CN disclosed
CN-113121427-A Quinoline derivative and preparation method and application thereof 广东工业大学 2021-07-16 CN disclosed