SCHEMBL28596643

SCHEMBL28596643

NC(=O)Oc1ccc(C=O)c([N+](=O)[O-])c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ERN1 O75460 8/20 0.43
ALDH1A1 P00352 5/20 0.43
MAPT P10636 3/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP3A4 P08684 1/20 0.43
ALOX15 P16050 1/20 0.43
PRKDC P78527 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ALDH5A1 P51649 1/20 0.37
ABAT P80404 1/20 0.37
PTGS2 P35354 1/20 0.37
MITF O75030 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
CCR6 P51684 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29197218 0.87 KDM4E (0.43) MEN1KMT2AALDH1A1MAPTKDM4E
SCHEMBL13779864 0.85 MAPT (0.46) MEN1KMT2AERN1ALDH1A1MAPT
SCHEMBL5693941 0.80 LMNA (0.54) MEN1KMT2AALDH1A1MAPTCYP3A4
SCHEMBL29269278 0.80 MAPK1 (0.54) MEN1KMT2AALDH1A1MAPTKDM4E
SCHEMBL23275859 0.78 MAPT (0.49) MEN1KMT2AALDH1A1MAPTKDM4E
SCHEMBL7161701 0.78 ALDH1A1 (0.50) MEN1KMT2AALDH1A1MAPTKDM4E
SCHEMBL28683817 0.78 VCAM1 (0.54) MEN1KMT2AALDH1A1MAPTCYP3A4
SCHEMBL1572278 0.78 ALDH1A1 (0.60) ERN1ALDH1A1MAPTKDM4ECYP3A4
SCHEMBL20958154 0.75 MAPT (0.45) MEN1KMT2AERN1ALDH1A1MAPT
SCHEMBL28474988 0.75 TSHR (0.53) MEN1KMT2AALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108250199-B Dihydropyridone P1 as factor XIA inhibitor 百时美施贵宝公司 2021-07-16 CN disclosed