SCHEMBL28599526

SCHEMBL28599526

O=C(O)C1CN(C(=O)c2cc(OCc3ccccc3)c(OCc3ccccc3)c(OCc3ccccc3)c2)CCN1S(=O)(=O)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.47
ALDH1A1 P00352 2/20 0.45
HSP90AA1 P07900 1/20 0.45
KMT2A Q03164 1/20 0.45
POLB P06746 1/20 0.44
HTT P42858 1/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA4 P22748 2/20 0.43
CA9 Q16790 2/20 0.43
MMP1 P03956 3/20 0.43
MMP3 P08254 3/20 0.43
MMP7 P09237 3/20 0.43
MMP9 P14780 3/20 0.43
MMP13 P45452 3/20 0.43
CYP19A1 P11511 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28618887 0.90 PTGES (0.46) PTGESALDH1A1HSP90AA1KMT2AMMP1
SCHEMBL28618883 0.84 PTGES (0.47) PTGESALDH1A1HSP90AA1KMT2APOLB
SCHEMBL28402624 0.82 NPC1 (0.58) PTGESALDH1A1KMT2APOLBHTT
SCHEMBL28919583 0.78 PTGES (0.46) PTGESALDH1A1HSP90AA1KMT2APOLB
SCHEMBL28599278 0.77 PTGES (0.45) PTGESALDH1A1HSP90AA1KMT2APOLB
SCHEMBL28402744 0.76 LMNA (0.54) ALDH1A1KMT2AHTT
SCHEMBL28400696 0.74 LMNA (0.60) ALDH1A1KMT2APOLBHTT
SCHEMBL28862339 0.73 PTGES (0.56) PTGESALDH1A1KMT2AHTTNPC1
SCHEMBL28397138 0.73 ALDH1A1 (0.59) ALDH1A1KMT2APOLBNPC1RAB9A
SCHEMBL28236192 0.71 GLRA1 (0.51) ALDH1A1KMT2APOLBCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113105395-B 4-phenylsulfonyl-1-trihydroxy benzoyl piperazine-2-carboxamide derivative and preparation method and application thereof 山东大学 2022-06-17 CN disclosed
CN-113105395-A 4-phenylsulfonyl-1-trihydroxy benzoyl piperazine-2-carboxamide derivative and preparation method and application thereof 山东大学 2021-07-13 CN disclosed