SCHEMBL28618883

SCHEMBL28618883

O=C(O)C1CN(S(=O)(=O)c2ccc([N+](=O)[O-])cc2)CCN1C(=O)c1cc(OCc2ccccc2)c(OCc2ccccc2)c(OCc2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.47
ALDH1A1 P00352 3/20 0.46
HSP90AA1 P07900 1/20 0.46
KMT2A Q03164 1/20 0.46
POLB P06746 1/20 0.45
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA4 P22748 2/20 0.43
CA9 Q16790 2/20 0.43
CYP19A1 P11511 3/20 0.42
FAAH O00519 2/20 0.40
HTT P42858 2/20 0.40
ADAM17 P78536 1/20 0.40
LMNA P02545 1/20 0.40
FOLH1 Q04609 1/20 0.39
MGLL Q99685 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28919583 0.92 PTGES (0.46) PTGESALDH1A1HSP90AA1KMT2APOLB
SCHEMBL28599278 0.91 PTGES (0.45) PTGESALDH1A1HSP90AA1KMT2APOLB
SCHEMBL28601960 0.89 CA1 (0.47) ALDH1A1KMT2APOLBCA1CA2
SCHEMBL28599526 0.84 PTGES (0.47) PTGESALDH1A1HSP90AA1KMT2APOLB
SCHEMBL28618887 0.77 PTGES (0.46) PTGESALDH1A1HSP90AA1KMT2ACYP19A1
SCHEMBL28402624 0.76 NPC1 (0.58) PTGESALDH1A1KMT2APOLBCA1
SCHEMBL28402744 0.75 LMNA (0.54) ALDH1A1KMT2AHTTLMNA
SCHEMBL28400696 0.73 LMNA (0.60) ALDH1A1KMT2APOLBHTTLMNA
SCHEMBL28606683 0.72 SPHK2 (0.42) CA1CA2CA4CA9
SCHEMBL1380872 0.69 ALDH1A1 (0.45) ALDH1A1HSP90AA1KMT2APOLBCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113105395-A 4-phenylsulfonyl-1-trihydroxy benzoyl piperazine-2-carboxamide derivative and preparation method and application thereof 山东大学 2021-07-13 CN claimed
CN-113105395-B 4-phenylsulfonyl-1-trihydroxy benzoyl piperazine-2-carboxamide derivative and preparation method and application thereof 山东大学 2022-06-17 CN disclosed
CN-113105395-A 4-phenylsulfonyl-1-trihydroxy benzoyl piperazine-2-carboxamide derivative and preparation method and application thereof 山东大学 2021-07-13 CN disclosed