SCHEMBL28599674

SCHEMBL28599674

O=C(Nc1ccc2ccccc2c1Br)c1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.66
RAB9A P51151 4/20 0.66
CYP1A2 P05177 1/20 0.66
CYP3A4 P08684 1/20 0.66
CYP2D6 P10635 1/20 0.66
CYP2C9 P11712 1/20 0.66
CYP2C19 P33261 1/20 0.66
MAPT P10636 3/20 0.50
KMT2A Q03164 5/20 0.49
MEN1 O00255 4/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
KCNJ11 Q14654 1/20 0.49
HDAC1 Q13547 2/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
MDM4 O15151 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28599669 0.85 MAPT (0.59) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL22798955 0.85 IMPDH2 (0.50) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL28613064 0.84 HDAC2 (0.57) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL9400456 0.82 NPC1 (0.68) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL777068 0.82 NPC1 (0.68) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL7478284 0.80 RXFP1 (0.60) NPC1RAB9AMAPTKMT2AMEN1
SCHEMBL31152642 0.80 RXFP1 (0.60) NPC1RAB9AMAPTKMT2AMEN1
SCHEMBL30184438 0.80 NPC1 (1.00) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL4642544 0.80 NPC1 (1.00) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL22532077 0.78 NPC1 (0.54) NPC1RAB9ACYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113200873-B Ortho-position halogenated arylamine compound and synthesis method thereof 山东硅科新材料有限公司 2023-02-03 CN disclosed
CN-113200873-A Ortho-position halogenated arylamine compound and synthesis method thereof 山东硅科新材料有限公司 2021-08-03 CN disclosed