SCHEMBL28600042

SCHEMBL28600042

CC(C)Cn1cc(C=O)c2cc(C#N)ccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.41
PFKFB2 O60825 3/20 0.39
PFKFB1 P16118 3/20 0.39
PFKFB3 Q16875 3/20 0.39
KMT2A Q03164 1/20 0.39
NR1D1 P20393 1/20 0.38
ICMT O60725 1/20 0.38
DPP4 P27487 2/20 0.38
GABRP O00591 1/20 0.37
GABRD O14764 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB1 P18505 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
GABRA2 P47869 1/20 0.37
GABRB2 P47870 1/20 0.37
GABRA4 P48169 1/20 0.37
GABRE P78334 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28597875 0.87 XDH (0.43) XDHICMTHTR3AKDM4EALDH1A1
SCHEMBL28592168 0.83 ICMT (0.42) ICMTHTR3AKDM4EALDH1A1GAA
SCHEMBL28587924 0.81 ALDH1A1 (0.39) XDHKMT2AGABRPGABRDGABRA1
SCHEMBL28613228 0.80 NR3C1 (0.40) XDHKMT2AGABRPGABRDGABRA1
SCHEMBL4350898 0.80 PTGER4 (0.43) KMT2AICMTKDM4EALDH1A1GAA
SCHEMBL28606673 0.80 SMN1; SMN2 (0.48) XDHKMT2AALDH1A1
SCHEMBL31346918 0.79 PTGDR2 (0.51) KMT2AKDM4EALDH1A1GAA
SCHEMBL28602068 0.78 ALDH1A1 (0.52) KMT2AALDH1A1
SCHEMBL13132153 0.78 NPC1 (0.50) ALDH1A1
SCHEMBL5440329 0.77 ALDH1A1 (0.60) KMT2AGABRPGABRDGABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113173917-B 1-alkyl-5-tetrazolyl/pyrimidone-1H-indole-3-carbonitrile compound and preparation method and application thereof 沈阳药科大学 2022-04-08 CN disclosed
CN-113173917-A 1-alkyl-5-tetrazolyl/pyrimidone-1H-indole-3-carbonitrile compound and preparation method and application thereof 沈阳药科大学 2021-07-27 CN disclosed