SCHEMBL28601933

SCHEMBL28601933

CC(NC(=O)c1noc(-c2ccccc2)n1)c1ccccc1Cl

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.58
HDAC6 Q9UBN7 3/20 0.58
HDAC8 Q9BY41 2/20 0.58
SMPD1 P17405 1/20 0.44
TSHR P16473 1/20 0.43
MAPK3 P27361 1/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 2/20 0.42
S1PR1 P21453 1/20 0.42
S1PR3 Q99500 1/20 0.42
MEN1 O00255 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
ROCK2 O75116 4/20 0.41
ROCK1 Q13464 3/20 0.41
TDP1 Q9NUW8 1/20 0.41
THRB P10828 1/20 0.41
PDE2A O00408 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28606427 0.79 TDP1 (0.51) MAPK3MAPK1KMT2AS1PR1S1PR3
SCHEMBL28608113 0.79 HDAC1 (0.56) HDAC1HDAC6HDAC8MAPK3MAPK1
SCHEMBL28597828 0.77 PTPN1 (0.48) HDAC6SMPD1MAPK3MAPK1L3MBTL1
SCHEMBL2104880 0.75 HDAC6 (0.77) HDAC1HDAC6HDAC8SMPD1TSHR
SCHEMBL28601974 0.74 MEN1 (0.61) MAPK3MAPK1KMT2AMEN1ROCK2
SCHEMBL28598671 0.73 CTSA (0.59) MAPK3MAPK1KMT2AMEN1ROCK2
SCHEMBL28601931 0.72 HDAC1 (0.59) HDAC1HDAC6HDAC8SMPD1TSHR
SCHEMBL2559848 0.72 HDAC6 (0.77) HDAC1HDAC6HDAC8SMPD1TSHR
SCHEMBL28611023 0.71 TUBB4A (0.50) HDAC1HDAC6HDAC8MAPK3MAPK1
SCHEMBL14959517 0.70 HDAC6 (0.68) HDAC1HDAC6HDAC8SMPD1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110407824-B Aryl formamide compound and preparation method, pharmaceutical composition and application thereof 安徽医科大学 2021-07-02 CN disclosed