SCHEMBL28602452

SCHEMBL28602452

Brc1cccc2[nH]cc(-c3ncco3)c12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 7/20 0.56
CDK5R1 Q15078 7/20 0.56
CLK1 P49759 6/20 0.56
CYP2A6 P11509 1/20 0.42
FGFR1 P11362 2/20 0.40
FGFR2 P21802 2/20 0.40
FGFR3 P22607 2/20 0.40
GSK3B P49841 3/20 0.37
HTR1A P08908 2/20 0.37
HTR2B P41595 2/20 0.37
CCNB2 O95067 2/20 0.37
CDK1 P06493 2/20 0.37
CCNB1 P14635 2/20 0.37
PRKACA P17612 2/20 0.37
PRKACG P22612 2/20 0.37
PRKACB P22694 2/20 0.37
CCNB3 Q8WWL7 2/20 0.37
PDPK1 O15530 1/20 0.37
CCNT1 O60563 1/20 0.37
CCNA2 P20248 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28613532 0.82 GPR84 (0.44) CDK5CDK5R1CLK1GSK3BHTR1A
SCHEMBL1352370 0.75 IMPDH2 (0.51) CDK5CDK5R1CLK1GSK3BHTR2B
SCHEMBL4739891 0.72 BRD4 (0.45) ADRA1DADRA1ABRD4HPGDS
SCHEMBL22053014 0.70 BRD4 (0.38) ADRA1DADRA1ABRD4CYP1B1HPGDS
SCHEMBL13544531 0.69 CLK1 (0.50) CDK5CDK5R1CLK1CYP2A6FGFR1
SCHEMBL7573578 0.68 ADRA1A (0.36) ADRA1DADRA1ABRD4CYP1B1HPGDS
SCHEMBL29197589 0.68 IMPDH2 (0.50) CDK5CDK5R1CLK1GSK3BHTR2B
SCHEMBL28973447 0.67 CYP2A6 (0.60) CDK5CDK5R1CLK1CYP2A6FGFR1
SCHEMBL26259967 0.66 BRD4 (0.53) ADRA1DADRA1ABRD4CYP1B1HPGDS
SCHEMBL1919495 0.65 HPGDS (0.52) ADRA1DADRA1ABRD4HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113185503-B Natural product Pimpirinine derivative and preparation method and application thereof 南京农业大学 2023-02-28 CN disclosed
CN-113185503-A Natural product Pimpirinine derivative and preparation method and application thereof 南京农业大学 2021-07-30 CN disclosed