SCHEMBL28604136

SCHEMBL28604136

NC(=O)OC1CCN(Cc2c[nH]c3ncc(Br)cc23)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 5/20 0.42
DRD2 P14416 4/20 0.39
DRD4 P21917 4/20 0.39
DRD3 P35462 4/20 0.39
SIGMAR1 Q99720 1/20 0.39
KRAS P01116 1/20 0.37
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
JAK1 P23458 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CYP2D6 P10635 1/20 0.36
JAK2 O60674 2/20 0.36
TYK2 P29597 2/20 0.36
JAK3 P52333 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16913887 0.78 LMNA (0.44) DRD2DRD4DRD3SIGMAR1KMT2A
SCHEMBL30007952 0.75 DRD4 (0.59) DRD2DRD4DRD3SIGMAR1MEN1
SCHEMBL30007886 0.75 GFER (0.47) DRD2DRD4DRD3SIGMAR1KMT2A
SCHEMBL29215986 0.75 EGFR (0.47) DRD2DRD4DRD3SIGMAR1KMT2A
SCHEMBL30008538 0.74 ALDH1A1 (0.41) DRD2DRD4DRD3JAK1KMT2A
SCHEMBL25296328 0.72 PLK4 (0.44) JAK2JAK3GAAPDPK1
SCHEMBL25303627 0.68 AURKA (0.49) JAK2JAK3KDM4EALDH1A1LMNA
SCHEMBL22864675 0.67 PDPK1 (0.52) JAK2JAK3KDM4EALDH1A1LMNA
SCHEMBL28541244 0.67 SCD (0.41) KDM4E
SCHEMBL5339464 0.67 SPR (0.55) BCHEACHEKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113121531-B N-heteroindole compound, synthesis method and medical application thereof 上海药明康德新药开发有限公司 2023-06-13 CN disclosed
CN-113121531-A N-heteroindole compound, and synthesis method and medical application thereof 上海药明康德新药开发有限公司 2021-07-16 CN disclosed