SCHEMBL30007952

SCHEMBL30007952

Brc1cnc2[nH]cc(CN3CCC(c4ccccc4)CC3)c2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 8/20 0.59
DRD2 P14416 6/20 0.59
DRD3 P35462 6/20 0.59
PLK4 O00444 1/20 0.46
AURKA O14965 1/20 0.46
JAK2 O60674 1/20 0.46
ROCK2 O75116 1/20 0.46
PRKD3 O94806 1/20 0.46
MAP4K4 O95819 1/20 0.46
PRKCG P05129 1/20 0.46
INSR P06213 1/20 0.46
CDK1 P06493 1/20 0.46
FES P07332 1/20 0.46
IGF1R P08069 1/20 0.46
ROS1 P08922 1/20 0.46
FGFR1 P11362 1/20 0.46
PHKG2 P15735 1/20 0.46
FER P16591 1/20 0.46
FLT1 P17948 1/20 0.46
CDK2 P24941 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16913887 0.81 LMNA (0.44) DRD4DRD2DRD3PLK4AURKA
SCHEMBL30007886 0.77 GFER (0.47) DRD4DRD2DRD3PLK4AURKA
SCHEMBL29215986 0.77 EGFR (0.47) DRD4DRD2DRD3PLK4AURKA
SCHEMBL30007369 0.76 DRD2 (0.47) DRD4DRD2DRD3INSRCDK2
SCHEMBL30008538 0.76 ALDH1A1 (0.41) DRD4DRD2DRD3HTR2AKMT2A
SCHEMBL28604136 0.75 SOS1 (0.42) DRD4DRD2DRD3JAK2JAK3
SCHEMBL29204307 0.70 MAP4K1 (0.64) PLK4AURKAJAK2ROCK2PRKD3
SCHEMBL22619026 0.69 DRD2 (0.87) DRD4DRD2DRD3JAK2KMT2A
SCHEMBL31326340 0.69 MPO (0.47) DRD4DRD2DRD3PLK4AURKA
SCHEMBL31326325 0.69 HTR2A (0.48) DRD4DRD2DRD3PLK4AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022237922-A1 ANTITUMOR COMPOUNDS BASED ON NITROGEN HETEROCYCLES AND USE THEREOF AS MEDICAMENTS FAKULTNI NEMOCNICE HRADEC KRALOVE (CZ) 2022-11-17 WO disclosed