SCHEMBL286047

SCHEMBL286047

CCCCc1noc(C)c1C=Cc1ncc(C(=O)OCC(N)=O)s1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.34
DBF4 Q9UBU7 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
KDM4E B2RXH2 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
ALDH1A1 P00352 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL286257 0.84 PRKAB2 (0.38) L3MBTL1KDM4ETDP1ALDH1A1SMN1; SMN2
SCHEMBL286258 0.84 PRKAB2 (0.38) L3MBTL1KDM4ETDP1ALDH1A1SMN1; SMN2
SCHEMBL286008 0.82 ALDH1A1 (0.35) L3MBTL1ALDH1A1SMN1; SMN2
SCHEMBL286010 0.82 ALDH1A1 (0.35) L3MBTL1ALDH1A1SMN1; SMN2
SCHEMBL285784 0.82 TSHR (0.35) CDC7DBF4L3MBTL1KDM4EALDH1A1
SCHEMBL286009 0.79 POLB (0.37) L3MBTL1KDM4EALDH1A1SMN1; SMN2
SCHEMBL286104 0.79 POLB (0.44) L3MBTL1CYP2D6CYP2C9CYP2C19TDP1
SCHEMBL286228 0.79 ALDH1A1 (0.36) CDC7DBF4L3MBTL1CYP2C9CYP2C19
SCHEMBL285969 0.78 STAT3 (0.35) KDM4EALDH1A1SMN1; SMN2
SCHEMBL286049 0.76 GABRA5 (0.43) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427459-A1 ISOXAZOLE-THIAZOLE DERIVATIVES AS GABA A RECEPTOR INVERSE AGONISTS FOR USE IN THE TREATMENT OF COGNITIVE DISORDERS F. Hoffmann-La Roche AG (CH) 2012-03-14 EP disclosed