SCHEMBL2860573

SCHEMBL2860573

CC(C)(C)[S@@+]([O-])NCCc1ccc(C(F)(F)F)nc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 3/20 0.41
TKT P29401 1/20 0.38
TRPV4 Q9HBA0 1/20 0.38
KDM1A O60341 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
CYP3A4 P08684 1/20 0.35
CYP3A5 P20815 1/20 0.35
PLAAT3 P53816 1/20 0.35
PLAAT5 Q96KN8 1/20 0.35
PLAAT2 Q9NWW9 1/20 0.35
PLAAT4 Q9UL19 1/20 0.35
EP300 Q09472 1/20 0.35
PPARD Q03181 1/20 0.33
KCNQ3 O43525 1/20 0.33
KCNQ2 O43526 1/20 0.33
KCNQ4 P56696 1/20 0.33
KCNQ5 Q9NR82 1/20 0.33
CYP2C19 P33261 1/20 0.33
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2860576 1.00 DAO (0.41) DAOTKTTRPV4KDM1AMAOA
SCHEMBL29162108 0.85 KDM1A (0.44) DAOTKTTRPV4KDM1AMAOA
SCHEMBL17981985 0.81 LOXL2 (0.48) KCNQ2
SCHEMBL16935058 0.79 HRH3 (0.34) CYP3A4KCNH2
SCHEMBL22265161 0.76 CARM1 (0.43) MAOBCYP2C19KCNH2
Hydrochloric Acid SCHEMBL20582040 0.74 DAO (0.46) DAOTKTTRPV4KDM1AMAOA
SCHEMBL2466202 0.74 DAO (0.46) DAOTKTTRPV4KDM1AMAOA
SCHEMBL1134880 0.73 NFKB1 (0.34) CYP3A4
SCHEMBL16516003 0.73 PTGS2 (0.31)
SCHEMBL16516002 0.73 PTGS2 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139334-A1 2-CYANOPHENYL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF Renovis, Inc. (US) 2010-01-06 EP disclosed
EP-2136639-A1 PYRID-2-YL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF Renovis, Inc. (US) 2009-12-30 EP disclosed
WO-2008130481-A1 2-CYANOPHENYL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF RENOVIS, INC. (US) 2008-10-30 WO disclosed
WO-2008123963-A1 PYRID-2-YL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF RENOVIS, INC. (US) 2008-10-16 WO disclosed