SCHEMBL28607232

SCHEMBL28607232

Clc1ccc2oc(Sc3nc(Cl)cc(Cl)n3)nc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.50
LMNA P02545 5/20 0.50
MAPK1 P28482 4/20 0.50
KDM4E B2RXH2 3/20 0.50
CYP1A2 P05177 2/20 0.50
TP53 P04637 2/20 0.50
HSD17B10 Q99714 2/20 0.50
ALDH1A1 P00352 2/20 0.50
RAB9A P51151 2/20 0.50
NPSR1 Q6W5P4 2/20 0.50
THRB P10828 1/20 0.50
ALOX15 P16050 1/20 0.50
S1PR2 O95136 1/20 0.50
XBP1 P17861 1/20 0.50
TMEM97 Q5BJF2 3/20 0.47
POLB P06746 1/20 0.47
CYP2C19 P33261 1/20 0.47
PSMB8 P28062 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
CASP3 P42574 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29594002 1.00 MAPT (0.50) MAPTLMNAMAPK1KDM4ECYP1A2
SCHEMBL28597642 0.85 LMNA (0.38) MAPTLMNAMAPK1KDM4ECYP1A2
SCHEMBL28597503 0.85 RAB9A (0.45) MAPTLMNAMAPK1KDM4ETP53
SCHEMBL29593441 0.85 MAPT (0.40) MAPTLMNAMAPK1KDM4ECYP1A2
SCHEMBL29593143 0.85 RAB9A (0.45) MAPTLMNAMAPK1KDM4ETP53
SCHEMBL29593098 0.85 LMNA (0.38) MAPTLMNAMAPK1KDM4ECYP1A2
SCHEMBL28597499 0.85 MAPT (0.40) MAPTLMNAMAPK1KDM4ECYP1A2
SCHEMBL28609798 0.83 MAPT (0.50) MAPTLMNAMAPK1KDM4ETP53
SCHEMBL28597508 0.82 FBP1 (0.43) MAPTLMNAMAPK1KDM4ETP53
SCHEMBL29593022 0.82 FBP1 (0.43) MAPTLMNAMAPK1KDM4ETP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113185511-B Pyrimidine compound and preparation method and application thereof 中国医学科学院医药生物技术研究所 2022-04-26 CN disclosed
CN-113185511-A Pyrimidine compound and preparation method and application thereof 中国医学科学院医药生物技术研究所 2021-07-30 CN disclosed