SCHEMBL28611181

SCHEMBL28611181

CN(C(=O)C1CN(S(=O)(=O)c2ccc(C#N)cc2)CCN1C(=O)c1cc(O)c(O)c(O)c1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA4 P22748 2/20 0.40
CA9 Q16790 2/20 0.40
ALDH1A1 P00352 2/20 0.38
ADAM17 P78536 1/20 0.37
KMT2A Q03164 1/20 0.37
F2 P00734 1/20 0.37
F10 P00742 1/20 0.37
OPRK1 P41145 1/20 0.36
PAX8 Q06710 1/20 0.36
GBA1 P04062 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PKM P14618 1/20 0.35
PKLR P30613 1/20 0.35
MMP8 P22894 2/20 0.35
MMP3 P08254 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28617316 0.89 CA1 (0.43) GAACA1CA2CA4CA9
SCHEMBL29720620 0.83 F10 (0.41) GAACA1CA2CA4CA9
SCHEMBL28618855 0.83 MAPT (0.46) GAACA1CA2CA4CA9
SCHEMBL28618201 0.76 F2 (0.44) GAACA1CA2CA4CA9
SCHEMBL28618856 0.75 ALDH1A1 (0.56) GAAALDH1A1KMT2AL3MBTL1PKM
SCHEMBL28608791 0.74 HTT (0.47) GAAADAM17PKMMMP3
SCHEMBL3714114 0.74 PDK2 (0.49) GAACA1CA2CA4CA9
SCHEMBL3709524 0.74 PDK2 (0.49) GAACA1CA2CA4CA9
SCHEMBL28608723 0.72 MMP1 (0.45) GAACA1CA2CA4CA9
SCHEMBL3721437 0.71 CA1 (0.56) GAACA1CA2CA4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113105395-B 4-phenylsulfonyl-1-trihydroxy benzoyl piperazine-2-carboxamide derivative and preparation method and application thereof 山东大学 2022-06-17 CN disclosed
CN-113105395-A 4-phenylsulfonyl-1-trihydroxy benzoyl piperazine-2-carboxamide derivative and preparation method and application thereof 山东大学 2021-07-13 CN disclosed