SCHEMBL28617316

SCHEMBL28617316

CN(C(=O)C1CN(S(=O)(=O)c2ccc(N)cc2)CCN1C(=O)c1cc(O)c(O)c(O)c1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.43
CA2 P00918 4/20 0.43
CA4 P22748 4/20 0.43
CA9 Q16790 4/20 0.43
GAA P10253 2/20 0.42
ALDH1A1 P00352 3/20 0.39
KMT2A Q03164 3/20 0.38
F2 P00734 1/20 0.38
F10 P00742 1/20 0.38
OPRK1 P41145 1/20 0.38
ADAM17 P78536 1/20 0.37
MEN1 O00255 2/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28611181 0.89 GAA (0.40) CA1CA2CA4CA9GAA
SCHEMBL28608723 0.83 MMP1 (0.45) CA1CA2CA4CA9GAA
SCHEMBL29720703 0.83 CA2 (0.43) CA1CA2CA4CA9ALDH1A1
SCHEMBL28611268 0.82 CA1 (0.44) CA1CA2CA4CA9GAA
SCHEMBL28604351 0.74 PKM (0.48) GAAALDH1A1
SCHEMBL28599524 0.74 ALDH1A1 (0.58) GAAALDH1A1KMT2AMEN1TDP1
SCHEMBL28601239 0.73 HTT (0.49) GAAALDH1A1KMT2A
SCHEMBL29720620 0.72 F10 (0.41) CA1CA2CA4CA9GAA
SCHEMBL28618855 0.71 MAPT (0.46) CA1CA2CA4CA9GAA
SCHEMBL7893587 0.69 CA1 (0.62) CA1CA2CA4CA9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113105395-B 4-phenylsulfonyl-1-trihydroxy benzoyl piperazine-2-carboxamide derivative and preparation method and application thereof 山东大学 2022-06-17 CN disclosed
CN-113105395-A 4-phenylsulfonyl-1-trihydroxy benzoyl piperazine-2-carboxamide derivative and preparation method and application thereof 山东大学 2021-07-13 CN disclosed