SCHEMBL28612072

SCHEMBL28612072

CCC(=O)N(c1ccccc1)C1CCN(c2ccccc2CN2CCN(OC(=O)C(C)(C)C)CC2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 11/20 0.54
SIGMAR1 Q99720 2/20 0.54
OPRD1 P41143 2/20 0.48
CHRM3 P20309 2/20 0.48
SLC22A1 O15245 1/20 0.48
NR1I2 O75469 1/20 0.48
ABCB1 P08183 1/20 0.48
CHRM1 P11229 1/20 0.48
DRD2 P14416 1/20 0.48
ADRA2B P18089 1/20 0.48
ADRA2C P18825 1/20 0.48
MAOA P21397 1/20 0.48
DRD4 P21917 1/20 0.48
MAOB P27338 1/20 0.48
ADRA1A P35348 1/20 0.48
HRH1 P35367 1/20 0.48
ADRA1B P35368 1/20 0.48
DRD3 P35462 1/20 0.48
OPRK1 P41145 1/20 0.48
CHRNA4 P43681 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28627150 0.89 OPRM1 (0.50) OPRM1SIGMAR1OPRD1CHRM3SLC22A1
SCHEMBL28613846 0.86 OPRM1 (0.55) OPRM1SIGMAR1OPRD1CHRM3SLC22A1
SCHEMBL28619729 0.82 OPRM1 (0.61) OPRM1SIGMAR1OPRD1CHRM3SLC22A1
SCHEMBL30632150 0.82 OPRM1 (0.61) OPRM1SIGMAR1OPRD1CHRM3SLC22A1
SCHEMBL27588773 0.81 OPRM1 (0.64) OPRM1SIGMAR1OPRD1CHRM3SLC22A1
Tert-Butyl Formate SCHEMBL28612074 0.80 OPRM1 (0.52) OPRM1SIGMAR1OPRD1CHRM3SLC22A1
SCHEMBL28616266 0.78 OPRM1 (0.49) OPRM1SIGMAR1OPRD1CHRM3SLC22A1
SCHEMBL30632148 0.78 OPRM1 (0.49) OPRM1SIGMAR1OPRD1CHRM3SLC22A1
SCHEMBL28627152 0.76 MGLL (0.53) OPRM1SIGMAR1MEN1KMT2A
SCHEMBL30632138 0.76 SMN1; SMN2 (0.52) OPRM1SIGMAR1OPRD1CHRM3SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113292485-A Benzylpiperazine urea TRPV1 antagonistic and MOR agonistic double-target-point medicine, preparation method and application 河南大学 2021-08-24 CN disclosed