SCHEMBL28612430

SCHEMBL28612430

Cc1ccc2c(c1)C(=O)CC(c1ccccc1)N2.NNC(=O)Nc1ccc(Br)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
BCL2 P10415 1/20 0.36
BECN1 Q14457 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
TP53 P04637 1/20 0.36
THRB P10828 1/20 0.36
FPR2 P25090 2/20 0.35
FPR1 P21462 1/20 0.35
EPHX2 P34913 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28603932 0.94 ALDH1A1 (0.39) NPC1RAB9ASMN1; SMN2TP53THRB
SCHEMBL28612434 0.92 MAPT (0.42) RAB9ASMN1; SMN2TP53FPR2FPR1
SCHEMBL28601605 0.89 KDR (0.39) MAOAMAOBNPC1RAB9ASMN1; SMN2
SCHEMBL28603992 0.89 KDR (0.39) MAOAMAOBNPC1RAB9ASMN1; SMN2
SCHEMBL28606070 0.89 GRIK1 (0.42) MAOAMAOBNPC1RAB9AHCRTR1
SCHEMBL28598799 0.89 IDH1 (0.38) NPC1RAB9ASMN1; SMN2TP53FPR2
SCHEMBL28598858 0.89 IDH1 (0.38) NPC1RAB9ASMN1; SMN2TP53FPR2
Aza-Flavanone SCHEMBL28606333 0.88 MAOA (0.45) MAOAMAOBSMN1; SMN2HCRTR1HCRTR2
SCHEMBL28612665 0.87 ALDH1A1 (0.40) NPC1RAB9ASMN1; SMN2FPR2FPR1
Aza-Flavanone SCHEMBL28608106 0.86 KDR (0.42) NPC1RAB9ASMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108558756-B 2-aryl-2, 3-dihydro-4 (1H) -quinolinone semicarbazone compound and application thereof 沈阳药科大学 2021-08-03 CN claimed