SCHEMBL28601605

SCHEMBL28601605

Cc1ccc(C2CC(=O)c3ccccc3N2)cc1.NNC(=O)Nc1ccc(Br)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
MAPT P10636 3/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CYP2C9 P11712 1/20 0.37
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
FPR1 P21462 1/20 0.36
POLB P06746 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
RECQL P46063 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28603992 1.00 KDR (0.39) KDRMAOAMAOBMAPTNPC1
SCHEMBL28919461 0.95 MAOA (0.42) MAOAMAOBMAPTNPC1RAB9A
Aza-Flavanone SCHEMBL28606333 0.93 MAOA (0.45) MAOAMAOBMAPTHCRTR1HCRTR2
Aza-Flavanone SCHEMBL28608106 0.93 KDR (0.42) KDRMAPTNPC1RAB9AMEN1
SCHEMBL28603909 0.90 KDR (0.40) KDRMAOAMAOBMAPTNPC1
SCHEMBL28614837 0.90 KDR (0.40) KDRMAOAMAOBMAPTNPC1
SCHEMBL28919462 0.89 FPR1 (0.48) RAB9AMEN1KMT2ATNKS2FPR1
SCHEMBL28601602 0.89 FPR1 (0.48) RAB9AMEN1KMT2ATNKS2FPR1
SCHEMBL28604164 0.89 GAA (0.42) KDRMAPTNPC1RAB9AMEN1
SCHEMBL28612430 0.89 MAOA (0.40) MAOAMAOBNPC1RAB9AHCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108558756-B 2-aryl-2, 3-dihydro-4 (1H) -quinolinone semicarbazone compound and application thereof 沈阳药科大学 2021-08-03 CN claimed