SCHEMBL28613166

SCHEMBL28613166

O=C(O)N1CCOc2ncccc2C1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 3/20 0.38
CREBBP Q92793 1/20 0.38
GPR142 Q7Z601 2/20 0.37
RIPK1 Q13546 2/20 0.37
HPGD P15428 3/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HSD17B10 Q99714 1/20 0.36
NAMPT P43490 2/20 0.36
SHMT2 P34897 1/20 0.35
HSD11B1 P28845 1/20 0.35
GAA P10253 1/20 0.35
LMNA P02545 1/20 0.35
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
GRM5 P41594 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3793892 0.87 LTA4H (0.39) PIK3CACREBBPGPR142RIPK1HPGD
SCHEMBL2113016 0.80 MAPK1 (0.53) NAMPTGRM5
SCHEMBL21800527 0.79 RIPK1 (0.62) RIPK1
SCHEMBL2111759 0.75 ABHD6 (0.40) PIK3CAGPR142RIPK1HPGDNAMPT
SCHEMBL17957763 0.75 RIPK1 (0.54) PIK3CAGPR142RIPK1HPGDKDM4E
SCHEMBL21710240 0.75 MAOA (0.43) LMNA
SCHEMBL29501124 0.75 RIPK1 (0.54) PIK3CAGPR142RIPK1HPGDKDM4E
SCHEMBL30895944 0.75 AHR (0.67) KDM4EALDH1A1GAALMNAGRM5
SCHEMBL20305088 0.74 PIK3CA (0.39) PIK3CACREBBPGPR142RIPK1NAMPT
SCHEMBL30314393 0.74 RIPK1 (0.49) RIPK1HPGDKDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137557-B Nrf2 modulators 葛兰素史密斯克莱知识产权发展有限公司 2021-09-07 CN disclosed