SCHEMBL28613328

SCHEMBL28613328

COC(=O)c1nsc(Br)c1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.43
KDM4E B2RXH2 9/20 0.36
ALDH1A1 P00352 6/20 0.36
HPGD P15428 4/20 0.36
HSD17B10 Q99714 4/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
PKM P14618 3/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
TP53 P04637 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
STAT3 P40763 1/20 0.33
HIF1A Q16665 1/20 0.33
MAPT P10636 2/20 0.33
RCE1 Q9Y256 2/20 0.33
TSHR P16473 2/20 0.33
NPC1 O15118 1/20 0.33
MAPK1 P28482 1/20 0.33
RAB9A P51151 1/20 0.33
GLA P06280 2/20 0.33
GAA P10253 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4756836 0.72 NPSR1 (0.45) NPSR1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL1549089 0.70 ALDH1A1 (0.54) NPSR1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL28627797 0.68 KDM4E (0.63) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL28623297 0.68 IKBKB (0.47) NPSR1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL17885172 0.68 KDM4E (0.40) NPSR1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL20049782 0.68 ALDH1A1 (0.57) NPSR1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL15872816 0.68 NPSR1 (0.50) NPSR1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL29790146 0.68 ALDH1A1 (0.46) NPSR1KDM4EALDH1A1HPGDL3MBTL1
SCHEMBL25290051 0.67 NPSR1 (0.54) NPSR1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9296458 0.67 NPSR1 (0.48) NPSR1KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118108744-A Isothiazolopyrimidinone compounds, pharmaceutical compositions containing the same and uses thereof 四川科伦博泰生物医药股份有限公司 2024-05-31 CN disclosed
CN-113087724-B Isothiazolopyrimidinone compounds, pharmaceutical compositions containing the same and uses thereof 四川科伦博泰生物医药股份有限公司 2024-01-19 CN disclosed
CN-113087724-A Isothiazolopyrimidinones, pharmaceutical compositions containing the same and uses thereof 四川科伦博泰生物医药股份有限公司 2021-07-09 CN disclosed