SCHEMBL28614161

SCHEMBL28614161

CC(C)(C)NC(=O)O[C@@H]1CCCN(c2ncc(OCC(F)(F)F)cc2Cl)C1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACACB O00763 5/20 0.45
SMN1; SMN2 Q16637 4/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
LMNA P02545 3/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
PRCP P42785 1/20 0.39
CNR2 P34972 2/20 0.39
CTSS P25774 1/20 0.39
CXCR3 P49682 1/20 0.38
GAA P10253 1/20 0.38
KDM4E B2RXH2 1/20 0.38
CNR1 P21554 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28607375 0.94 ACACB (0.50) ACACBSMN1; SMN2MEN1KMT2ALMNA
SCHEMBL28614142 0.87 SMN1; SMN2 (0.53) SMN1; SMN2MEN1KMT2ALMNAALDH1A1
SCHEMBL28605624 0.87 SMN1; SMN2 (0.53) SMN1; SMN2MEN1KMT2ALMNAALDH1A1
SCHEMBL28595526 0.86 GPR119 (0.45) ACACBSMN1; SMN2MEN1KMT2ALMNA
SCHEMBL28595527 0.86 GPR119 (0.45) ACACBSMN1; SMN2MEN1KMT2ALMNA
SCHEMBL28605601 0.85 NTMT1 (0.42) ACACBSMN1; SMN2MEN1KMT2ALMNA
SCHEMBL28610083 0.83 MEN1 (0.38) SMN1; SMN2MEN1KMT2ALMNAALDH1A1
SCHEMBL28614165 0.81 BTK (0.51) ACACBMEN1KMT2A
SCHEMBL31124450 0.81 BTK (0.51) ACACBMEN1KMT2A
SCHEMBL28614149 0.80 MEN1 (0.43) ACACBSMN1; SMN2MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113164461-A Heterocyclic derivatives as Nav1.7 and Nav1.8 blockers 拉夸里亚创药株式会社 2021-07-23 CN disclosed