SCHEMBL28617167

SCHEMBL28617167

Nc1nn(CC(F)(F)F)c2cccc(Cl)c12

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.36
KDR P35968 1/20 0.36
ESR1 P03372 1/20 0.36
GAA P10253 2/20 0.36
MAPK14 Q16539 1/20 0.36
CYP17A1 P05093 2/20 0.35
IL1B P01584 2/20 0.34
P2RX7 Q99572 2/20 0.34
RORC P51449 4/20 0.33
CNR1 P21554 1/20 0.33
PIK3CD O00329 1/20 0.32
SRC P12931 1/20 0.32
TOP2A P11388 1/20 0.31
PRMT5 O14744 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17038937 0.79 NR1H2 (0.43) P2RX7RORC
SCHEMBL30695004 0.79 NR1H2 (0.43) P2RX7RORC
SCHEMBL17199358 0.76 RORC (0.36) GAARORC
SCHEMBL10372436 0.74 GAA (0.35) GAARORCCNR1TOP2A
SCHEMBL21420031 0.73 NOTUM (0.33) RETKDR
SCHEMBL19875661 0.73 RET (0.33) RETKDR
SCHEMBL13241454 0.72 ABHD6 (0.43) CNR1
SCHEMBL23439990 0.71 P2RX7 (0.34) RETKDRMAPK14P2RX7
SCHEMBL23993155 0.70 CNR1 (0.43) MAPK14CYP17A1RORCCNR1
SCHEMBL23994521 0.69 HTR3A (0.42) RETKDRESR1CYP17A1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113195475-A Inhibitors of human immunodeficiency virus replication VIIV保健英国第五有限公司 2021-07-30 CN disclosed