SCHEMBL28619892

SCHEMBL28619892

NC(CCCc1ccccc1)C(F)(F)C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.44
MAOA P21397 1/20 0.42
MAOB P27338 2/20 0.41
HTR2A P28223 1/20 0.41
FAAH O00519 3/20 0.40
CES1 P23141 3/20 0.40
IDO1 P14902 1/20 0.40
S1PR2 O95136 1/20 0.39
S1PR4 O95977 1/20 0.39
S1PR1 P21453 1/20 0.39
S1PR3 Q99500 1/20 0.39
ANPEP P15144 2/20 0.39
ERAP1 Q9NZ08 2/20 0.39
ERAP2 Q6P179 1/20 0.39
SIGMAR1 Q99720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28615047 0.89 ANPEP (0.44) MAOAMAOBHTR2ACES1IDO1
SCHEMBL3488301 0.75 FAAH (0.50) MAOAMAOBFAAHCES1S1PR2
SCHEMBL5789705 0.74 MAOA (0.54) GRIK1MAOAMAOBHTR2AIDO1
SCHEMBL3266047 0.74 S1PR2 (0.59) GRIK1MAOAMAOBHTR2AIDO1
SCHEMBL5807580 0.74 GRIK1 (0.46) GRIK1MAOAMAOBHTR2AFAAH
SCHEMBL7953179 0.73 ANPEP (0.47) MAOAMAOBHTR2AIDO1ANPEP
Hydrochloric Acid SCHEMBL10535805 0.72 MAOB (0.54) GRIK1MAOAMAOBHTR2AIDO1
Hydrochloric Acid SCHEMBL1979100 0.72 S1PR2 (0.57) GRIK1MAOAMAOBHTR2AIDO1
SCHEMBL14544283 0.71 GRIK1 (0.54) GRIK1MAOAMAOBHTR2AIDO1
SCHEMBL3712834 0.71 SLC6A2 (0.56) GRIK1MAOAMAOBHTR2ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107949562-B Positive allosteric modulators of muscarinic M2 receptors 拜耳制药股份公司 2021-07-23 CN disclosed